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Cat. No. Product Name Target Signaling Pathways
T9911 Tocilizumab

Interleukin Immunology/Inflammation
Tocilizumab 是抗人白细胞介素-6 受体 (IL-6R) 的中和抗体,能够阻碍 IL-6 与 IL-6R 的结合,进而抑制经典和反式信号。它可用于研究类风湿性关节炎,对重症 COVID-19 冠状病毒病方面的研究具有显著效果。
TP1016L Aviptadil Acetate

醋酸阿肽地尔,阿肽地尔,Vasoactive Intestinal Peptide acetate salt

RAAS; SARS-CoV Endocrinology/Hormones; Microbiology/Virology
Aviptadil Acetate (Vasoactive Intestinal Peptide acetate salt) 是模拟血管活性肠多肽类似物,具有血管舒张效应。它可诱导肺血管舒张并抑制血管 SMC 的增殖和血小板聚集。它可用于研究 SARS-CoV-2 引起的肺纤维化、肺动脉高压和呼吸衰竭。
T76690 Mavrilimumab

CAM 3001

Virus Protease; CSF-1R Microbiology/Virology; Tyrosine Kinase/Adaptors
Mavrilimumab (CAM 3001) 是一种单克隆抗体,具有抗病毒活性,对粒细胞-巨噬细胞集落刺激因子 (GM-CSF) 受体的 α 亚基有亲和力,并阻止 GM-CSF 下游细胞内信号传导。GM-CSF 可能与呼吸衰竭和死亡相关的过度活跃炎症反应有关,可用于研究类风湿性关节炎。
T21414 Sivelestat sodium

ONO 5046,LY-544349,Sivelestat sodium salt,ONO-5046,ONO5046,西维来司钠,LY544349,LY 544349

Sivelestat, an inhibitor of human neutrophil elastase, is used in the treatment of acute respiratory failure. Preliminary studies show Sivelestat may improve neuropathic pain.
T69786 GSK3491943

GSK3491943 is a potent TRPV4 inhibitor with IC50 = 3.2 nM. GSK3491943 is a potential agent for the treatment of heart failure and respiratory diseases.
T69784 GSK3527497 HCl

GSK3527497 is a potent and selective inhibitor of Transient Receptor Potential Vanilloid‑4 (TRPV4) with IC50 = 12 nM) for the treatment of heart failure and respiratory diseases. GSK3527497 is a preclinical candidate suitable for oral and iv administration that is projected to inhibit TRPV4 effectively in patients from a low daily clinical dose.

化合物

Tocilizumab
Cat.No: T9911
Synonym:
Target: Interleukin
Aviptadil Acetate
Cat.No: TP1016L
Synonym: 醋酸阿肽地尔,阿肽地尔,Vasoactive Intestinal Peptide acetate salt
Target: RAAS, SARS-CoV
Mavrilimumab
Cat.No: T76690
Synonym: CAM 3001
Target: Virus Protease, CSF-1R
Sivelestat sodium
Cat.No: T21414
Synonym: ONO 5046,LY-544349,Sivelestat sodium salt,ONO-5046,ONO5046,西维来司钠,LY544349,LY 544349
Target:
GSK3491943
Cat.No: T69786
Synonym:
Target:
GSK3527497 HCl
Cat.No: T69784
Synonym:
Target:
TargetMol Loading
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